1 |
Ramajayam_2010 |
Synthesis, docking studies, and evaluation of pyrimidines as inhibitors of SARS-CoV 3CL protease |
Ramajayam, R.; Tan, Kian-Pin; Liu, Hun-Ge; Liang, Po-Huang |
2010 |
2010-06-15 |
PMC |
N |
PMC7126861 |
20494577.0 |
10.1016/j.bmcl.2010.04.118 |
4g5dur1n |
0.902068 |
Ramajayam_2010, Regnier_2009 |
Konno_2017, Dude_2008, Regnier_2009, Duque_2009 |
2 |
Regnier_2009 |
New developments for the design, synthesis and biological evaluation of potent SARS-CoV 3CLpro inhibitors |
Regnier, Thomas; Sarma, Diganta; Hidaka, Koushi; Bacha, Usman; Freire, Ernesto; Hayashi, Yoshio; Kiso, Yoshiaki |
2009 |
2009-05-15 |
None |
N |
PMC4436079 |
19362479.0 |
10.1016/j.bmcl.2009.03.118 |
zxganumj |
0.882540 |
Ramajayam_2010, Ramajayam_2010, Chen_2005, Konno_2016 |
Ramajayam_2010, Konno_2017, Konno_2013, Konno_2016 |
3 |
Ohnishi_2019 |
Evaluation of a non-prime site substituent and warheads combined with a decahydroisoquinolin scaffold as a SARS 3CL protease inhibitor |
Ohnishi, Kouji; Hattori, Yasunao; Kobayashi, Kazuya; Akaji, Kenichi |
2019 |
2019-01-15 |
PMC |
N |
PMC7126642 |
30558861.0 |
10.1016/j.bmc.2018.12.019 |
960th627 |
0.841105 |
|
Yoshizawa_2020, Konno_2013, Thanigaimalai_2013 |
4 |
Yoshizawa_2020 |
Evaluation of an octahydroisochromene scaffold used as a novel SARS 3CL protease inhibitor |
Yoshizawa, Shin-ichiro; Hattori, Yasunao; Kobayashi, Kazuya; Akaji, Kenichi |
2020 |
2020-02-15 |
PMC |
N |
PMC7127348 |
31926775.0 |
10.1016/j.bmc.2019.115273 |
c5m4dj9m |
0.780829 |
|
Konno_2013, Pomeisl_2019, Thanigaimalai_2013 |
5 |
Lin_S_2020 |
Molecular Modeling Evaluation of the Binding Effect of Ritonavir, Lopinavir and Darunavir to Severe Acute Respiratory Syndrome Coronavirus 2 Proteases |
Shen Lin; Runnan Shen; Jingdong He; Xinhao Li; Xushun Guo |
2020 |
2020-02-03 |
BioRxiv |
Y |
|
|
10.1101/2020.01.31.929695 |
vbgf50os |
0.747112 |
|
Saijo_2005 |
6 |
Ramajayam_2010 |
Synthesis and evaluation of pyrazolone compounds as SARS-coronavirus 3C-like protease inhibitors |
Ramajayam, R.; Tan, Kian-Pin; Liu, Hun-Ge; Liang, Po-Huang |
2010 |
2010-11-15 |
PMC |
N |
PMC7127448 |
20947359.0 |
10.1016/j.bmc.2010.09.050 |
2keibgne |
0.735936 |
Ramajayam_2010, Regnier_2009 |
Ramajayam_2010, Konno_2016, Dude_2008, Chen_2005 |
7 |
Deaton_2008 |
Thiol-based angiotensin-converting enzyme 2 inhibitors: P1 modifications for the exploration of the S1 subsite |
Deaton, David N.; Gao, Enoch N.; Graham, Kevin P.; Gross, Jeffrey W.; Miller, Aaron B.; Strelow, John M. |
2008 |
2008-01-15 |
PMC |
N |
PMC7126659 |
18078750.0 |
10.1016/j.bmcl.2007.11.048 |
gic43uwz |
0.729478 |
Ramajayam_2010 |
Dude_2008 |
8 |
Shi_Y_2018 |
Identification of two antiviral inhibitors targeting 3C-like serine/3C-like protease of porcine reproductive and respiratory syndrome virus and porcine epidemic diarrhea virus |
Shi, Yuejun; Lei, Yingying; Ye, Gang; Sun, Limeng; Fang, Liurong; Xiao, Shaobo; Fu, Zhen F.; Yin, Ping; Song, Yunfeng; Peng, Guiqing |
2018 |
2018-01-31 |
PMC |
N |
PMC7117380 |
29291994.0 |
10.1016/j.vetmic.2017.11.031 |
ikjjjn4s |
0.708666 |
|
Hu_H_2019 |
9 |
Konno_2017 |
Synthesis and evaluation of phenylisoserine derivatives for the SARS-CoV 3CL protease inhibitor |
Konno, Hiroyuki; Onuma, Takumi; Nitanai, Ikumi; Wakabayashi, Masaki; Yano, Shigekazu; Teruya, Kenta; Akaji, Kenichi |
2017 |
2017-06-15 |
PMC |
N |
PMC7127027 |
28454669.0 |
10.1016/j.bmcl.2017.04.056 |
qym6jch0 |
0.674965 |
Ramajayam_2010 |
Ramajayam_2010, Konno_2016, Dude_2008, Konno_2013 |
10 |
Shie_2005 |
Inhibition of the severe acute respiratory syndrome 3CL protease by peptidomimetic α,β-unsaturated esters |
Shie, Jiun-Jie; Fang, Jim-Min; Kuo, Tun-Hsun; Kuo, Chih-Jung; Liang, Po-Huang; Huang, Hung-Jyun; Wu, Yin-Ta; Jan, Jia-Tsrong; Cheng, Yih-Shyun E.; Wong, Chi-Huey |
2005 |
2005-09-01 |
PMC |
N |
PMC7119063 |
15994085.0 |
10.1016/j.bmc.2005.05.065 |
9fiqf6lk |
0.670048 |
Ramajayam_2010 |
|
11 |
Sun_Y_2013 |
Synthesis and Biological Evaluation of Quinolinone Compounds as SARS CoV 3CL(pro) Inhibitors |
Sun, Yuanpei; Zhang, Ning; Wang, Jian; Guo, Yu; Sun, Bo; Liu, Wei; Zhou, Honggang; Yang, Cheng |
2013 |
2013-07-19 |
PMC |
N |
PMC7159103 |
|
10.1002/cjoc.201300392 |
ew6kqsfr |
0.655350 |
Ramajayam_2010 |
|
12 |
Konno_2016 |
Design and synthesis of a series of serine derivatives as small molecule inhibitors of the SARS coronavirus 3CL protease |
Konno, Hiroyuki; Wakabayashi, Masaki; Takanuma, Daiki; Saito, Yota; Akaji, Kenichi |
2016 |
2016-03-15 |
PMC |
N |
PMC7111485 |
26879854.0 |
10.1016/j.bmc.2016.01.052 |
9bw1z5ps |
0.609871 |
Ramajayam_2010, Regnier_2009, Ramajayam_2010 |
Dude_2008, Im_I_2009, Ramajayam_2010, Chen_2005 |
13 |
Konno_2013 |
Design and synthesis of new tripeptide-type SARS-CoV 3CL protease inhibitors containing an electrophilic arylketone moiety |
Konno, Sho; Thanigaimalai, Pillaiyar; Yamamoto, Takehito; Nakada, Kiyohiko; Kakiuchi, Rie; Takayama, Kentaro; Yamazaki, Yuri; Yakushiji, Fumika; Akaji, Kenichi; Kiso, Yoshiaki; Kawasaki, Yuko; Chen, Shen-En; Freire, Ernesto; Hayashi, Yoshio |
2013 |
2013-01-15 |
PMC |
N |
PMC7127713 |
23245752.0 |
10.1016/j.bmc.2012.11.017 |
esogd26s |
0.601624 |
|
Thanigaimalai_2013, Thanigaimalai_2013 |
14 |
Kumar_2016 |
Identification, synthesis and evaluation of SARS-CoV and MERS-CoV 3C-like protease inhibitors |
Kumar, Vathan; Tan, Kian-Pin; Wang, Ying-Ming; Lin, Sheng-Wei; Liang, Po-Huang |
2016 |
2016-07-01 |
PMC |
N |
PMC7079562 |
27240464.0 |
10.1016/j.bmc.2016.05.013 |
s9wb9275 |
0.594739 |
|
Liu_W_2014 |
15 |
Liu_W_2014 |
Synthesis, modification and docking studies of 5-sulfonyl isatin derivatives as SARS-CoV 3C-like protease inhibitors |
Liu, Wei; Zhu, He-Min; Niu, Guo-Jun; Shi, En-Zhi; Chen, Jie; Sun, Bo; Chen, Wei-Qiang; Zhou, Hong-Gang; Yang, Cheng |
2014 |
2014-01-01 |
None |
N |
PMC7111328 |
24316352.0 |
10.1016/j.bmc.2013.11.028 |
r0h2zhj2 |
0.576316 |
Ramajayam_2010 |
|
16 |
Hilgenfeld_2006 |
Sometimes Intermediates Do the Job! |
Hilgenfeld, Rolf; Pumpor, Ksenia |
2006 |
2006-03-31 |
PMC |
N |
PMC7111035 |
16638527.0 |
10.1016/j.chembiol.2006.03.002 |
ij5sr88p |
0.570985 |
David_2013 |
Dude_2008 |
17 |
Kao_R_2004 |
Identification of Novel Small-Molecule Inhibitors of Severe Acute Respiratory Syndrome-Associated Coronavirus by Chemical Genetics |
Kao, Richard Y.; Tsui, Wayne H.W.; Lee, Terri S.W.; Tanner, Julian A.; Watt, Rory M.; Huang, Jian-Dong; Hu, Lihong; Chen, Guanhua; Chen, Zhiwei; Zhang, Linqi; He, Tian; Chan, Kwok-Hung; Tse, Herman; To, Amanda P.C.; Ng, Louisa W.Y.; Wong, Bonnie C.W.; Tsoi, Hoi-Wah; Yang, Dan; Ho, David D.; Yuen, Kwok-Yung |
2004 |
2004-09-30 |
PMC |
N |
PMC7128553 |
15380189.0 |
10.1016/j.chembiol.2004.07.013 |
jgtbp5r6 |
0.549904 |
|
|
18 |
Ryu_Y_2010 |
Biflavonoids from Torreya nucifera displaying SARS-CoV 3CLpro inhibition |
Ryu, Young Bae; Jeong, Hyung Jae; Kim, Jang Hoon; Kim, Young Min; Park, Ji-Young; Kim, Doman; Naguyen, Thi Thanh Hanh; Park, Su-Jin; Chang, Jong Sun; Park, Ki Hun; Rho, Mun-Chual; Lee, Woo Song |
2010 |
2010-11-15 |
PMC |
N |
PMC7126309 |
20934345.0 |
10.1016/j.bmc.2010.09.035 |
4x5l2h4d |
0.521688 |
Kuo_R_2009 |
Gondim_2019, Park_2017 |
19 |
Peters_2015 |
Design, synthesis and evaluation of a series of acyclic fleximer nucleoside analogues with anti-coronavirus activity |
Peters, Hannah L.; Jochmans, Dirk; de Wilde, Adriaan H.; Posthuma, Clara C.; Snijder, Eric J.; Neyts, Johan; Seley-Radtke, Katherine L. |
2015 |
2015-08-01 |
None |
N |
PMC4466200 |
26048809.0 |
10.1016/j.bmcl.2015.05.039 |
9o0mc3rd |
0.512761 |
|
Hamada_2013, Cho_A_2012 |
20 |
Prior_2013 |
Design, synthesis, and bioevaluation of viral 3C and 3C-like protease inhibitors |
Prior, Allan M.; Kim, Yunjeong; Weerasekara, Sahani; Moroze, Meghan; Alliston, Kevin R.; Uy, Roxanne Adeline Z.; Groutas, William C.; Chang, Kyeong-Ok; Hua, Duy H. |
2013 |
2013-12-01 |
None |
N |
PMC3863581 |
24125888.0 |
10.1016/j.bmcl.2013.09.070 |
ly8ibnju |
0.508130 |
|
Im_I_2009, Cho_A_2012, Dude_2008 |
21 |
Shin_2020 |
Identification of 6′-β-fluoro-homoaristeromycin as a potent inhibitor of chikungunya virus replication |
Shin, Young Sup; Jarhad, Dnyandev B.; Jang, Min Hwan; Kovacikova, Kristina; Kim, Gyudong; Yoon, Ji-seong; Kim, Hong-Rae; Hyun, Young Eum; Tipnis, Amol S.; Chang, Tong-Shin; van Hemert, Martijn J.; Jeong, Lak Shin |
2020 |
2020-02-01 |
None |
N |
PMC7115507 |
31841728.0 |
10.1016/j.ejmech.2019.111956 |
hu8dzbhk |
0.499983 |
|
Yoon_2019, Piotrowska_2019, Mehellou_2010 |
22 |
Ma_C_2020 |
Boceprevir, GC-376, and calpain inhibitors II, XII inhibit SARS-CoV-2 viral replication by targeting the viral main protease |
Chunlong Ma; Brett Hurst; Yanmei Hu; Tommy Szeto; Bart Tarbet; Jun Wang |
2020 |
2020-04-20 |
BioRxiv |
Y |
|
|
10.1101/2020.04.20.051581 |
047xpt2c |
0.495778 |
|
|
23 |
Thanigaimalai_2013 |
Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: Structure–activity relationship study |
Thanigaimalai, Pillaiyar; Konno, Sho; Yamamoto, Takehito; Koiwai, Yuji; Taguchi, Akihiro; Takayama, Kentaro; Yakushiji, Fumika; Akaji, Kenichi; Kiso, Yoshiaki; Kawasaki, Yuko; Chen, Shen-En; Naser-Tavakolian, Aurash; Schön, Arne; Freire, Ernesto; Hayashi, Yoshio |
2013 |
2013-07-31 |
None |
N |
PMC7115367 |
23747811.0 |
10.1016/j.ejmech.2013.05.005 |
2i6795ga |
0.491212 |
Ramajayam_2010 |
Thanigaimalai_2013, Konno_2013 |
24 |
Ghosh_2008 |
Design, synthesis and antiviral efficacy of a series of potent chloropyridyl ester-derived SARS-CoV 3CLpro inhibitors |
Ghosh, Arun K.; Gong, Gangli; Grum-Tokars, Valerie; Mulhearn, Debbie C.; Baker, Susan C.; Coughlin, Melissa; Prabhakar, Bellur S.; Sleeman, Katrina; Johnson, Michael E.; Mesecar, Andrew D. |
2008 |
2008-10-15 |
None |
N |
PMC2745596 |
18796354.0 |
10.1016/j.bmcl.2008.08.082 |
sx3g8uvc |
0.489329 |
Ramajayam_2010 |
Ramajayam_2010, Cho_A_2012, Pérez-Faginas_2011, Konno_2016 |
25 |
Chng_2004 |
Synthetic studies towards anti-SARS agents: application of an indium-mediated allylation of α-aminoaldehydes as the key step towards an intermediate |
Chng, Shu-Sin; Hoang, Truong-Giang; Wayne Lee, Wei-Woon; Tham, Mun-Pun; Ling, Hui Yvonne; Loh, Teck-Peng |
2004 |
2004-12-20 |
PMC |
N |
PMC7119068 |
|
10.1016/j.tetlet.2004.10.146 |
x8xntne7 |
0.482736 |
MacDonald_2012, Ramajayam_2010 |
Ramajayam_2010, Cho_A_2012, Lin_Z_2012 |
26 |
Park_2013 |
Dieckol, a SARS-CoV 3CLpro inhibitor, isolated from the edible brown algae Ecklonia cava |
Park, Ji-Young; Kim, Jang Hoon; Kwon, Jung Min; Kwon, Hyung-Jun; Jeong, Hyung Jae; Kim, Young Min; Kim, Doman; Lee, Woo Song; Ryu, Young Bae |
2013 |
2013-07-01 |
PMC |
N |
PMC7126891 |
23647823.0 |
10.1016/j.bmc.2013.04.026 |
3uhjmocf |
0.479988 |
David_2013 |
Dude_2008, Ramajayam_2010, Konno_2017, Im_I_2009 |
27 |
Shao_2008 |
Design, synthesis, and evaluation of trifluoromethyl ketones as inhibitors of SARS-CoV 3CL protease |
Shao, Yi-Ming; Yang, Wen-Bin; Kuo, Tun-Hsun; Tsai, Keng-Chang; Lin, Chun-Hung; Yang, An-Suei; Liang, Po-Huang; Wong, Chi-Huey |
2008 |
2008-04-15 |
PMC |
N |
PMC7127754 |
18329272.0 |
10.1016/j.bmc.2008.02.040 |
pgzogpa2 |
0.478259 |
Ramajayam_2010, Regnier_2009 |
Pérez-Faginas_2011, Ramajayam_2010, Prior_2013, Konno_2016 |
28 |
Chen_2005 |
Inhibition of SARS-CoV 3C-like Protease Activity by Theaflavin-3,3′-digallate (TF3) |
Chen, Chia-Nan; Lin, Coney P. C.; Huang, Kuo-Kuei; Chen, Wei-Cheng; Hsieh, Hsin-Pang; Liang, Po-Huang; Hsu, John T.-A. |
2005 |
2005-04-07 |
PMC |
N |
PMC1142193 |
15937562.0 |
10.1093/ecam/neh081 |
0svscbpu |
0.476564 |
|
|
29 |
Kim_J_2017 |
Antiviral escin derivatives from the seeds of Aesculus turbinata Blume (Japanese horse chestnut) |
Kim, Ji Won; Ha, Thi-Kim-Quy; Cho, Hyomoon; Kim, Eunhee; Shim, Sang Hee; Yang, Jun-Li; Oh, Won Keun |
2017 |
2017-07-01 |
PMC |
N |
PMC7127610 |
28527823.0 |
10.1016/j.bmcl.2017.05.022 |
84u3c33m |
0.475412 |
|
|
30 |
Wu_C_2006 |
Stable Benzotriazole Esters as Mechanism-Based Inactivators of the Severe Acute Respiratory Syndrome 3CL Protease |
Wu, Chung-Yi; King, Ke-Yung; Kuo, Chih-Jung; Fang, Jim-Min; Wu, Ying-Ta; Ho, Ming-Yi; Liao, Chung-Lin; Shie, Jiun-Jie; Liang, Po-Huang; Wong, Chi-Huey |
2006 |
2006-03-31 |
None |
N |
PMC7111201 |
16638531.0 |
10.1016/j.chembiol.2005.12.008 |
bfrozfvg |
0.453377 |
|
|
31 |
Saijo_2005 |
Inhibitory effect of mizoribine and ribavirin on the replication of severe acute respiratory syndrome (SARS)-associated coronavirus |
Saijo, Masayuki; Morikawa, Shigeru; Fukushi, Shuetsu; Mizutani, Tetsuya; Hasegawa, Hideki; Nagata, Noriyo; Iwata, Naoko; Kurane, Ichiro |
2005 |
2005-06-30 |
PMC |
N |
PMC7114120 |
15911031.0 |
10.1016/j.antiviral.2005.01.003 |
drrs2tc1 |
0.439616 |
|
|
32 |
Keyaerts_2007 |
Plant lectins are potent inhibitors of coronaviruses by interfering with two targets in the viral replication cycle |
Keyaerts, Els; Vijgen, Leen; Pannecouque, Christophe; Van Damme, Els; Peumans, Willy; Egberink, Herman; Balzarini, Jan; Van Ranst, Marc |
2007 |
2007-09-30 |
PMC |
N |
PMC7114093 |
17428553.0 |
10.1016/j.antiviral.2007.03.003 |
6qmckoo8 |
0.407764 |
|
|
33 |
Dai_W_2020 |
Structure-Based Design, Synthesis and Biological Evaluation of Peptidomimetic Aldehydes as a Novel Series of Antiviral Drug Candidates Targeting the SARS-CoV-2 Main Protease |
Wenhao Dai; Bing Zhang; Xia-Ming Jiang; Haixia Su; Jian Li; Yao Zhao; Xiong Xie; Zhenming Jin; Jingjing Peng; Fengjiang Liu; Chunpu Li; You Li; Fang Bai; Haofeng Wang; Xi Cheng; Xiaobo Cen; Shulei Hu; Xiuna Yang; Jiang Wang; Xiang Liu; Gengfu Xiao; Hualiang Jiang; Zihe Rao; Leike Zhang; Yechun Xu; Haitao Yang; Hong Liu |
2020 |
2020-03-28 |
BioRxiv |
Y |
|
|
10.1101/2020.03.25.996348 |
b4joa5tx |
0.405492 |
|
Konno_2013, Thanigaimalai_2013, Thanigaimalai_2013 |
34 |
Kim_B_2015 |
Benserazide, the first allosteric inhibitor of Coxsackievirus B3 3C protease |
Kim, Bo-Kyoung; Cho, Joong-Heui; Jeong, Pyeonghwa; Lee, Youngjin; Lim, Jia Jia; Park, Kyoung Ryoung; Eom, Soo Hyun; Kim, Yong-Chul |
2015 |
2015-07-08 |
PMC |
N |
PMC7094222 |
26022398.0 |
10.1016/j.febslet.2015.05.027 |
4szi4vyd |
0.400129 |
|
Zhong_2009 |
35 |
Thanigaimalai_2013 |
Development of potent dipeptide-type SARS-CoV 3CL protease inhibitors with novel P3 scaffolds: Design, synthesis, biological evaluation, and docking studies |
Thanigaimalai, Pillaiyar; Konno, Sho; Yamamoto, Takehito; Koiwai, Yuji; Taguchi, Akihiro; Takayama, Kentaro; Yakushiji, Fumika; Akaji, Kenichi; Chen, Shen-En; Naser-Tavakolian, Aurash; Schön, Arne; Freire, Ernesto; Hayashi, Yoshio |
2013 |
2013-10-31 |
None |
N |
PMC7115411 |
23994330.0 |
10.1016/j.ejmech.2013.07.037 |
olfpcndb |
0.400094 |
|
Konno_2013, Thanigaimalai_2013 |
36 |
Keyaerts_2004 |
Inhibition of SARS-coronavirus infection in vitro by S-nitroso-N-acetylpenicillamine, a nitric oxide donor compound |
Keyaerts, Els; Vijgen, Leen; Chen, Luni; Maes, Piet; Hedenstierna, Göran; Van Ranst, Marc |
2004 |
2004-07-31 |
PMC |
N |
PMC7128975 |
15234326.0 |
10.1016/j.ijid.2004.04.012 |
78xva8a0 |
0.398324 |
|
|
37 |
Hu_D_2007 |
Studies on the interactions of Ti-containing polyoxometalates (POMs) with SARS-CoV 3CLpro by molecular modeling |
Hu, Donghua; Shao, Chen; Guan, Wei; Su, Zhongmin; Sun, Jiazhong |
2007 |
2007-01-31 |
None |
N |
PMC7112571 |
17049610.0 |
10.1016/j.jinorgbio.2006.08.013 |
azosg1tt |
0.391429 |
|
Thanigaimalai_2013 |
38 |
Hsu_J_2004 |
Evaluation of metal-conjugated compounds as inhibitors of 3CL protease of SARS-CoV |
Hsu, John T.-A.; Kuo, Chih-Jung; Hsieh, Hsing-Pang; Wang, Yeau-Ching; Huang, Kuo-Kuei; Lin, Coney P.-C.; Huang, Ping-Fang; Chen, Xin; Liang, Po-Huang |
2004 |
2004-09-10 |
PMC |
N |
PMC7134601 |
15358550.0 |
10.1016/j.febslet.2004.08.015 |
8sc6nbqp |
0.383965 |
Ramajayam_2010 |
Liu_W_2014 |
39 |
Yoon_2019 |
Design, Synthesis, and Anti-RNA Virus Activity of 6′-Fluorinated-Aristeromycin Analogues |
Yoon, Ji-seong; Kim, Gyudong; Jarhad, Dnyandev B.; Kim, Hong-Rae; Shin, Young-Sup; Qu, Shuhao; Sahu, Pramod K.; Kim, Hea Ok; Lee, Hyuk Woo; Wang, Su Bin; Kong, Yun Jeong; Chang, Tong-Shin; Ogando, Natacha S.; Kovacikova, Kristina; Snijder, Eric J.; Posthuma, Clara C.; van Hemert, Martijn J.; Jeong, Lak Shin |
2019 |
2019-06-07 |
None |
N |
PMC7075649 |
31244113.0 |
10.1021/acs.jmedchem.9b00781 |
gfumqmku |
0.382911 |
|
Shin_2020, Obeid_2011 |
40 |
Wang_2017 |
Discovery of unsymmetrical aromatic disulfides as novel inhibitors of SARS-CoV main protease: Chemical synthesis, biological evaluation, molecular docking and 3D-QSAR study |
Wang, Li; Bao, Bo-Bo; Song, Guo-Qing; Chen, Cheng; Zhang, Xu-Meng; Lu, Wei; Wang, Zefang; Cai, Yan; Li, Shuang; Fu, Sheng; Song, Fu-Hang; Yang, Haitao; Wang, Jian-Guo |
2017 |
2017-09-08 |
PMC |
N |
PMC7115414 |
28624700.0 |
10.1016/j.ejmech.2017.05.045 |
mxnx4mmu |
0.381075 |
|
Liu_W_2014, Thanigaimalai_2013 |
41 |
Günther_2004 |
Application of real-time PCR for testing antiviral compounds against Lassa virus, SARS coronavirus and Ebola virus in vitro |
Günther, Stephan; Asper, Marcel; Röser, Christina; Luna, Luciano K.S.; Drosten, Christian; Becker-Ziaja, Beate; Borowski, Peter; Chen, Huan-Ming; Hosmane, Ramachandra S. |
2004 |
2004-09-30 |
PMC |
N |
PMC7126008 |
15451189.0 |
10.1016/j.antiviral.2004.05.001 |
wys8t1wi |
0.380576 |
|
Obeid_2011 |
42 |
Li_S_2005 |
Identification of natural compounds with antiviral activities against SARS-associated coronavirus |
Li, Shi-you; Chen, Cong; Zhang, Hai-qing; Guo, Hai-yan; Wang, Hui; Wang, Lin; Zhang, Xiang; Hua, Shi-neng; Yu, Jun; Xiao, Pei-gen; Li, Rong-song; Tan, Xuehai |
2005 |
2005-07-31 |
PMC |
N |
PMC7114104 |
15885816.0 |
10.1016/j.antiviral.2005.02.007 |
4s57ls6y |
0.376489 |
Ishag_2016 |
Chen_2005 |
43 |
Choi_2009 |
Antiviral activity of quercetin 7-rhamnoside against porcine epidemic diarrhea virus |
Choi, Hwa-Jung; Kim, Jin-Hee; Lee, Choong-Hwan; Ahn, Young-Joon; Song, Jae-Hyoung; Baek, Seung-Hwa; Kwon, Dur-Han |
2009 |
2009-01-31 |
PMC |
N |
PMC7114206 |
18992773.0 |
10.1016/j.antiviral.2008.10.002 |
ni7qfjk9 |
0.373000 |
|
Hu_H_2019 |
44 |
Zhang_2008 |
Aryl methylene ketones and fluorinated methylene ketones as reversible inhibitors for severe acute respiratory syndrome (SARS) 3C-like proteinase |
Zhang, Jianmin; Huitema, Carly; Niu, Chunying; Yin, Jiang; James, Michael N.G.; Eltis, Lindsay D.; Vederas, John C. |
2008 |
2008-10-31 |
PMC |
N |
PMC7112044 |
18295820.0 |
10.1016/j.bioorg.2008.01.001 |
tv5yyfak |
0.358868 |
Ramajayam_2010 |
Pomeisl_2019, Ikejiri_2007, Głowacka_2015 |
45 |
Kang_2015 |
Jubanines F–J, cyclopeptide alkaloids from the roots of Ziziphus jujuba |
Kang, Kyo Bin; Ming, Gao; Kim, Geum Jin; Ha, Thi-Kim-Quy; Choi, Hyukjae; Oh, Won Keun; Sung, Sang Hyun |
2015 |
2015-11-30 |
PMC |
N |
PMC7111685 |
26361730.0 |
10.1016/j.phytochem.2015.09.001 |
lib3slrw |
0.340366 |
David_2013 |
Li_X_2019 |
46 |
Lim_J_2020 |
The Author's Response: Case of the Index Patient Who Caused Tertiary Transmission of Coronavirus Disease 2019 in Korea: the Application of Lopinavir/Ritonavir for the Treatment of COVID-19 Pneumonia Monitored by Quantitative RT-PCR |
Lim, Jaegyun; Jeon, Seunghyun; Shin, Hyun Young; Kim, Moon Jung; Seong, Yu Min; Lee, Wang Jun; Choe, Kang Won; Kang, Yu Min; Lee, Baeckseung; Park, Sang Joon |
2020 |
2020-01-01 |
NONCOMM |
N |
|
32080993.0 |
10.3346/jkms.2020.35.e89 |
fjmchbew |
0.339476 |
|
|
47 |
David_2013 |
Ethyl dibromofluoroacetate: a versatile reagent for the synthesis of fluorinated molecules |
David, Emilie; Couve-Bonnaire, Samuel; Jubault, Philippe; Pannecoucke, Xavier |
2013 |
2013-12-30 |
PMC |
N |
PMC7126840 |
|
10.1016/j.tet.2013.10.048 |
xdihvg6k |
0.339476 |
|
Lin_Z_2012, Kale_2010 |
48 |
Shigeta_2006 |
Anti-RNA virus activity of polyoxometalates |
Shigeta, Shiro; Mori, Shuichi; Yamase, Toshihiro; Yamamoto, Norio; Yamamoto, Naoki |
2006 |
2006-06-30 |
PMC |
N |
PMC7118841 |
16737794.0 |
10.1016/j.biopha.2006.03.009 |
siyyve9e |
0.336535 |
|
|
49 |
Chen_2005 |
Synthesis and evaluation of isatin derivatives as effective SARS coronavirus 3CL protease inhibitors |
Chen, Li-Rung; Wang, Yu-Chin; Lin, Yi Wen; Chou, Shan-Yen; Chen, Shyh-Fong; Liu, Lee Tai; Wu, Ying-Ta; Kuo, Chih-Jung; Chen, Tom Shieh-Shung; Juang, Shin-Hun |
2005 |
2005-06-15 |
PMC |
N |
PMC7119080 |
15896959.0 |
10.1016/j.bmcl.2005.04.027 |
9he52hq5 |
0.333790 |
Ramajayam_2010, Regnier_2009, Ramajayam_2010, Konno_2016 |
Konno_2016, Dude_2008, Ramajayam_2010, Ramajayam_2010 |
50 |
Sydnes_2006 |
Synthesis of glutamic acid and glutamine peptides possessing a trifluoromethyl ketone group as SARS-CoV 3CL protease inhibitors |
Sydnes, Magne O.; Hayashi, Yoshio; Sharma, Vinay K.; Hamada, Takashi; Bacha, Usman; Barrila, Jennifer; Freire, Ernesto; Kiso, Yoshiaki |
2006 |
2006-09-04 |
None |
N |
PMC7111793 |
|
10.1016/j.tet.2006.06.052 |
mf0k7h27 |
0.333710 |
David_2013 |
Rauvolfova_2008, Głowacka_2015, Tsoukala_2010 |
51 |
Han_D_2006 |
Identification of critical determinants on ACE2 for SARS-CoV entry and development of a potent entry inhibitor |
Han, Dong P.; Penn-Nicholson, Adam; Cho, Michael W. |
2006 |
2006-06-20 |
PMC |
Y |
PMC7111894 |
16510163.0 |
10.1016/j.virol.2006.01.029 |
v1mf5lhh |
0.317044 |
|
|
52 |
Báez-Santos_2014 |
X-ray Structural and Biological Evaluation of a Series of Potent and Highly Selective Inhibitors of Human Coronavirus Papain-like Proteases |
Báez-Santos, Yahira\nM.; Barraza, Scott J.; Wilson, Michael W.; Agius, Michael P.; Mielech, Anna M.; Davis, Nicole M.; Baker, Susan C.; Larsen, Scott D.; Mesecar, Andrew D. |
2014 |
2014-02-25 |
PMC |
N |
PMC3983375 |
24568342.0 |
10.1021/jm401712t |
pkcsqnp4 |
0.311530 |
|
Thanigaimalai_2013, Konno_2013 |