1 |
Desai_2013 |
Synthesis, antimicrobial and cytotoxic activities of some novel thiazole clubbed 1,3,4-oxadiazoles |
Desai, N.C.; Bhatt, Nayan; Somani, Hardik; Trivedi, Amit |
2013 |
2013-09-30 |
PMC |
N |
PMC7127452 |
23835482.0 |
10.1016/j.ejmech.2013.06.029 |
mqcwk2ow |
0.966062 |
Mohammat_2009, Rajić_2010, Zhang_2018, Kuo_R_2009 |
Sahoo_2016, Zhong_2017, Cihan-Üstündağ_2019 |
2 |
Nadaraia_2018 |
Synthesis and Biological Activity of Several Modified 5α-Androstanolone Derivatives |
Nadaraia, N. Sh.; Barbakadze, N. N.; Kakhabrishvili, M. L.; Sylla, B.; Pichette, A.; Makhmudov, U. S. |
2018 |
2018-04-14 |
PMC |
N |
PMC7087839 |
|
10.1007/s10600-018-2330-2 |
ns32sje1 |
0.955832 |
Kuo_R_2009, Mohammat_2009, Regnier_2009 |
Duque_2009, Yadav_2005, Cho_A_2012 |
3 |
Balzarini_2014 |
Structural Analogs of Umifenovir. 1. Synthesis and Biological Activity of Ethyl 5-Hydroxy-1-Methyl-2-(Trans-2-Phenylcyclopropyl)-1H-Indole-3-Carboxylate |
Balzarini, J.; Ruchko, E. A.; Zakharova, E. K.; Kameneva, I. Yu.; Nawrozkij, M. B. |
2014 |
2014-06-08 |
PMC |
N |
PMC7088350 |
|
10.1007/s10593-014-1499-y |
2yhj3m9i |
0.937081 |
Kale_2010, Lin_Z_2012 |
Kumarapperuma_2007, Paramonova_2017, Duque_2009, Głowacka_2015 |
4 |
Yadav_2010 |
4-[1-(Substituted aryl/alkyl carbonyl)-benzoimidazol-2-yl]-benzenesulfonic acids: Synthesis, antimicrobial activity, QSAR studies, and antiviral evaluation |
Yadav, Snehlata; Kumar, Pradeep; De Clercq, Erik; Balzarini, Jan; Pannecouque, Christophe; Dewan, Sharwan Kumar; Narasimhan, Balasubramanian |
2010 |
2010-12-31 |
PMC |
N |
PMC7115694 |
20971531.0 |
10.1016/j.ejmech.2010.09.065 |
6jffpajp |
0.913563 |
|
Kumar_2014, Lakshman_2014, Sahoo_2016, Pomeisl_2019 |
5 |
Sahoo_2016 |
Antimicrobial activity of novel synthesized coumarin based transitional metal complexes |
Sahoo, Jyotirmaya; Paidesetty, Sudhir K. |
2016 |
2016-11-24 |
None |
N |
PMC6694993 |
31435225.0 |
10.1016/j.jtumed.2016.10.004 |
v4dje5yl |
0.862393 |
David_2013, Mohammat_2009 |
Pahonțu_2015, Carbone_2013, Pomeisl_2019 |
6 |
Kumar_2010 |
Benzylidene/2-chlorobenzylidene hydrazides: Synthesis, antimicrobial activity, QSAR studies and antiviral evaluation |
Kumar, Davinder; Judge, Vikramjeet; Narang, Rakesh; Sangwan, Sonia; De Clercq, Erik; Balzarini, Jan; Narasimhan, Balasubramanian |
2010 |
2010-07-31 |
PMC |
N |
PMC7127590 |
20347509.0 |
10.1016/j.ejmech.2010.03.002 |
e1sz07u3 |
0.845861 |
|
Sahoo_2016, Cihan-Üstündağ_2019, Desai_2013 |
7 |
Szűcs_2018 |
Structure-activity relationship studies of lipophilic teicoplanin pseudoaglycon derivatives as new anti-influenza virus agents |
Szűcs, Zsolt; Kelemen, Viktor; Le Thai, Son; Csávás, Magdolna; Rőth, Erzsébet; Batta, Gyula; Stevaert, Annelies; Vanderlinden, Evelien; Naesens, Lieve; Herczegh, Pál; Borbás, Anikó |
2018 |
2018-09-05 |
None |
N |
PMC7115582 |
30170320.0 |
10.1016/j.ejmech.2018.08.058 |
wclwpq7v |
0.839718 |
Singh_2013 |
McGuigan_2013, Mehellou_2010 |
8 |
Karaküçük-İyidoğan_2011 |
Novel platinum(II) and palladium(II) complexes of thiosemicarbazones derived from 5-substitutedthiophene-2-carboxaldehydes and their antiviral and cytotoxic activities |
Karaküçük-İyidoğan, Ayşegül; Taşdemir, Demet; Oruç-Emre, Emine Elçin; Balzarini, Jan |
2011 |
2011-11-30 |
PMC |
N |
PMC7126824 |
21993152.0 |
10.1016/j.ejmech.2011.09.031 |
cekegxop |
0.794368 |
Desai_2013, Mohammat_2009 |
Sahoo_2016, Pahonțu_2015, Thomson_2010, Cihan-Üstündağ_2019 |
9 |
Kumar_2014 |
Synthesis, antimicrobial, anticancer, antiviral evaluation and QSAR studies of 4-(1-aryl-2-oxo-1,2-dihydro-indol-3-ylideneamino)-N-substituted benzene sulfonamides |
Kumar, Mahesh; Ramasamy, Kalavathy; Mani, Vasudevan; Mishra, Rakesh Kumar; Majeed, Abu Bakar Abdul; Clercq, Erik De; Narasimhan, Balasubramanian |
2014 |
2014-09-30 |
PMC |
N |
|
|
10.1016/j.arabjc.2012.12.005 |
jys8vod1 |
0.783214 |
Desai_2013, Roman_2015 |
Sahoo_2016, Bari_2020, Carbone_2013 |
10 |
Mohammat_2009 |
Synthesis of 2,3-Dioxo-5-(substituted)arylpyrroles and Their 2-Oxo-5-aryl-3-hydrazone Pyrrolidine Derivatives |
Mohammat, M.F.; Shaameri, Z.; Hamzah, A.S. |
2009 |
2009-01-07 |
COMM-USE |
N |
PMC6253891 |
19136912.0 |
10.3390/molecules14010250 |
b9wq9gj6 |
0.755121 |
MacDonald_2012, Nadaraia_2018, Desai_2013, Desai_2013 |
Paramonova_2017, Tayade_2015, Riahi_2009, Pomeisl_2019 |
11 |
Sokolova_2013 |
New quaternary ammonium camphor derivatives and their antiviral activity, genotoxic effects and cytotoxicity |
Sokolova, Anastasiya S.; Yarovaya, Оlga I.; Shernyukov, Аndrey V.; Pokrovsky, Мichail A.; Pokrovsky, Аndrey G.; Lavrinenko, Valentina A.; Zarubaev, Vladimir V.; Tretiak, Tatiana S.; Anfimov, Pavel M.; Kiselev, Oleg I.; Beklemishev, Anatoly B.; Salakhutdinov, Nariman F. |
2013 |
2013-11-01 |
PMC |
N |
PMC7126328 |
23993669.0 |
10.1016/j.bmc.2013.08.014 |
2kytuxxy |
0.748511 |
|
Sahoo_2016, Gazivoda_2008 |
12 |
Hjortland_2016 |
Steady-state kinetic studies reveal that the anti-cancer target Ubiquitin-Specific Protease 17 (USP17) is a highly efficient deubiquitinating enzyme |
Hjortland, Nicole M.; Mesecar, Andrew D. |
2016 |
2016-12-01 |
PMC |
N |
PMC5868344 |
27756680.0 |
10.1016/j.abb.2016.10.008 |
nwl5i9h6 |
0.716192 |
|
|
13 |
Pomarnacka_2011 |
Synthesis, Cytotoxicity Testing, and Structure–Activity Relationships of Novel 6‐Chloro‐7‐(4‐phenylimino‐4H‐3,1‐benzoxazin‐2‐yl)‐3‐(substituted)‐1,4,2‐benzodithiazine 1,1‐dioxides |
Pomarnacka, Elżbieta; Kornicka, Anita; Kuchnio, Anna; Heinrichs, Maike; Grünert, Renate; Gdaniec, Maria; Bednarski, Patrick J. |
2011 |
2011-05-25 |
PMC |
N |
PMC7159733 |
21618270.0 |
10.1002/ardp.201000183 |
ahsyp92n |
0.714341 |
|
|
14 |
Desai_2013 |
Synthesis and antimicrobial activity of novel quinazolinone–thiazolidine–quinoline compounds |
Desai, N.C.; Dodiya, Amit; Shihory, Niraj |
2013 |
2013-07-31 |
PMC |
N |
PMC7148931 |
|
10.1016/j.jscs.2011.04.001 |
tndrp8dp |
0.705320 |
|
Sahoo_2016, Carbone_2013, Desai_2013 |
15 |
Kazakova_2011 |
Synthesis of a-secomethylenamino- and substituted amidoximotriterpenoids |
Kazakova, O. B.; Giniyatullina, G. V.; Tolstikov, G. A. |
2011 |
2011-10-01 |
PMC |
N |
PMC7088524 |
22332366.0 |
10.1134/s1068162011050086 |
ur15ywlr |
0.702193 |
MacDonald_2012, Mlostoń_2010, Kuo_R_2009, Yazarians_2017, Roman_2015 |
Kasthuri_2011, Chopade_2016, Tayade_2015, Paramonova_2017 |
16 |
Siddiqui_2011 |
Synthesis and anticonvulsant properties of 1-(amino-N-arylmethanethio)-3-(1-substituted benzyl-2, 3-dioxoindolin-5-yl) urea derivatives |
Siddiqui, Nadeem; Alam, M. Shamsher; Stables, James P. |
2011 |
2011-06-30 |
PMC |
N |
PMC7115639 |
21435751.0 |
10.1016/j.ejmech.2011.03.004 |
31e2db0z |
0.701881 |
Desai_2013, Duque_2009, Yadav_2005, Rajić_2010 |
Pomeisl_2019, Tsoukala_2010, Piotrowska_2012, Karki_2012 |
17 |
Hassan_2016 |
Therapeutic potential of coumarins as antiviral agents |
Hassan, Mohd. Zaheen; Osman, Hasnah; Ali, Mohamed Ashraf; Ahsan, Mohamed Jawed |
2016 |
2016-11-10 |
PMC |
N |
PMC7115672 |
27484512.0 |
10.1016/j.ejmech.2016.07.056 |
ahceohgl |
0.697476 |
|
Singh_2013 |
18 |
Kumar_2012 |
N′-[4-[(Substituted imino)methyl]benzylidene]-substituted benzohydrazides: synthesis, antimicrobial, antiviral, and anticancer evaluation, and QSAR studies |
Kumar, Pradeep; Narasimhan, Balasubramanian; Ramasamy, Kalavathy; Mani, Vasudevan; Mishra, Rakesh Kumar; Majeed, Abu Bakar Abdul; De Clercq, Erik |
2012 |
2012-12-01 |
PMC |
N |
PMC7087754 |
|
10.1007/s00706-012-0877-3 |
wf36hx8o |
0.693006 |
David_2013 |
Sahoo_2016, Kumar_2014, Pomeisl_2019 |
19 |
Ukrainets_2008 |
4-Hydroxy-2-quinolones 139. Synthesis, structure, and antiviral activity of N-R-amides of 2-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxylic acids |
Ukrainets, I. V.; Bereznyakova, N. L.; Turaibei, I. A. |
2008 |
2008-05-31 |
PMC |
N |
PMC7088292 |
|
10.1007/s10593-008-0012-x |
qe5w17iz |
0.660551 |
|
Paramonova_2017, Głowacka_2015, Kumarapperuma_2007 |
20 |
Gangarapu_2013 |
Synthesis of thiocarbohydrazide and carbohydrazide derivatives as possible biologically active agents |
Gangarapu, Kiran; Manda, Sarangapani; Jallapally, Anvesh; Thota, Sreekanth; Karki, Subhas S.; Balzarini, Jan; De Clercq, Erik; Tokuda, Harukuni |
2013 |
2013-08-23 |
PMC |
N |
PMC7080202 |
|
10.1007/s00044-013-0684-3 |
85xcc71l |
0.658691 |
David_2013, Mohammat_2009 |
Sahoo_2016, Chopade_2016, Carbone_2013 |
21 |
Novikov_2013 |
N1,N3-disubstituted uracils as nonnucleoside inhibitors of HIV-1 reverse transcriptase |
Novikov, Mikhail S.; Valuev-Elliston, Vladimir T.; Babkov, Denis A.; Paramonova, Maria P.; Ivanov, Alexander V.; Gavryushov, Sergey A; Khandazhinskaya, Anastasia L.; Kochetkov, Sergey N.; Pannecouque, Christophe; Andrei, Graciela; Snoeck, Robert; Balzarini, Jan; Seley-Radtke, Katherine L. |
2013 |
2013-03-01 |
PMC |
N |
PMC7125863 |
23357038.0 |
10.1016/j.bmc.2012.12.027 |
9bay2qaq |
0.655579 |
Novikov_2011 |
Cho_A_2012, Pérez-Faginas_2011, Im_I_2009 |
22 |
Torres_2010 |
Polycyclic N‐Benzamido Imides with Potent Activity against Vaccinia Virus |
Torres, Eva; Duque, María D.; Camps, Pelayo; Naesens, Lieve; Calvet, Teresa; Font‐Bardia, Mercè; Vázquez, Santiago |
2010 |
2010-10-21 |
None |
N |
PMC7162373 |
20967819.0 |
10.1002/cmdc.201000306 |
lj6przme |
0.649375 |
|
|
23 |
Zhao_2019 |
Research progress in the biological activities of 3,4,5-trimethoxycinnamic acid (TMCA) derivatives |
Zhao, Zefeng; Song, Huanhuan; Xie, Jing; Liu, Tian; Zhao, Xue; Chen, Xufei; He, Xirui; Wu, Shaoping; Zhang, Yongmin; Zheng, Xiaohui |
2019 |
2019-07-01 |
PMC |
N |
PMC7115657 |
31009908.0 |
10.1016/j.ejmech.2019.04.009 |
01mvhsrk |
0.646889 |
|
Bozorov_2019, Sahoo_2016 |
24 |
Seley-Radtke_2018 |
Flexibility—Not just for yoga anymore! |
Seley-Radtke, Katherine |
2018 |
2018-02-21 |
NONCOMM |
N |
PMC5890542 |
29466861.0 |
10.1177/2040206618756788 |
b6h9tw5o |
0.633903 |
|
|
25 |
More_2019 |
Metal complexes driven from Schiff bases and semicarbazones for biomedical and allied applications: a review |
More, M.S.; Joshi, P.G.; Mishra, Y.K.; Khanna, P.K. |
2019 |
2019-12-31 |
PMC |
N |
PMC7110249 |
|
10.1016/j.mtchem.2019.100195 |
p3ocduvi |
0.626433 |
Abu-Dief_2015, MacDonald_2012, Bozorov_2019 |
Abu-Dief_2015, Sahoo_2016, Bozorov_2019, Kryshchyshyn_2018 |
26 |
Rajić_2010 |
The novel amidocarbamate derivatives of ketoprofen: synthesis and biological activity |
Rajić, Zrinka; Hadjipavlou-Litina, Dimitra; Pontiki, Eleni; Balzarini, Jan; Zorc, Branka |
2010 |
2010-02-03 |
PMC |
N |
PMC7079954 |
|
10.1007/s00044-010-9309-2 |
90wgik7n |
0.619649 |
David_2013 |
Sahoo_2016, Piotrowska_2019, Pomeisl_2019, Carbone_2013 |
27 |
Kumbar_2020 |
Anticancer activity studies of novel metal complexes of ligands derived from polycyclic aromatic compound via greener route |
Kumbar, Mahantesh; Patil, Sangamesh A.; Toragalmath, Shivakumar S.; Kinnal, Shivashankar M.; Shettar, Arun; Hosakeri, Joy H. |
2020 |
2020-03-07 |
PMC |
N |
|
|
10.1016/j.jorganchem.2020.121219 |
2frdhhnm |
0.616517 |
Mohammat_2009 |
Sahoo_2016, More_2019, Carbone_2013, Pahonțu_2015 |
28 |
Pervez_2011 |
Synthesis and Toxicity Evaluation of Some N(4)-Aryl Substituted 5-Trifluoromethoxyisatin-3-thiosemicarbazones |
Pervez, Humayun; Saira, Naveeda; Iqbal, Mohammad Saeed; Yaqub, Muhammad; Khan, Khalid Mohammed |
2011 |
2011-07-29 |
COMM-USE |
N |
PMC6264754 |
25134761.0 |
10.3390/molecules16086408 |
a7hiw0vw |
0.614074 |
David_2013 |
Pomeisl_2019, Głowacka_2015, Głowacka_2016, Carbone_2013 |
29 |
Paramonova_2017 |
Novel 1-[5-(4-bromophenoxy)pentyl]-3-(2-arylamino- 2-oxoethyl)uracils and their antiviral properties |
Paramonova, Maria P.; Khandazhinskaya, Anastasia L.; Seley-Radtke, Katherine L.; Novikov, Mikhail S. |
2017 |
2017-02-28 |
PMC |
N |
|
|
10.1016/j.mencom.2017.01.027 |
sfl5nrc4 |
0.608149 |
Singh_2013, Mohammat_2009 |
Riahi_2009, Tayade_2015, Mohammat_2009, Novikov_2013 |
30 |
Park_2012 |
Synthesis and antiviral evaluation of 7-O-arylmethylquercetin derivatives against SARS-associated coronavirus (SCV) and hepatitis C virus (HCV) |
Park, Hye Ri; Yoon, Hyunjun; Kim, Mi Kyoung; Lee, Sung Dae; Chong, Youhoon |
2012 |
2012-02-02 |
PMC |
N |
PMC7090976 |
22297745.0 |
10.1007/s12272-012-0108-9 |
59bqlc5y |
0.596587 |
|
Ikejiri_2007, Kim_M_2011, Zhong_2015 |
31 |
Lee_C_2009 |
Investigation of the pharmacophore space of Severe Acute Respiratory Syndrome coronavirus (SARS-CoV) NTPase/helicase by dihydroxychromone derivatives |
Lee, Chaewoon; Lee, Jin Moo; Lee, Na-Ra; Kim, Dong-Eun; Jeong, Yong-Joo; Chong, Youhoon |
2009 |
2009-08-15 |
PMC |
N |
PMC7127646 |
19625187.0 |
10.1016/j.bmcl.2009.07.009 |
texnuvvp |
0.594654 |
|
|
32 |
Abu-Dief_2015 |
A review on versatile applications of transition metal complexes incorporating Schiff bases |
Abu-Dief, Ahmed M.; Mohamed, Ibrahim M.A. |
2015 |
2015-06-30 |
PMC |
N |
PMC7104041 |
|
10.1016/j.bjbas.2015.05.004 |
65r3pkqi |
0.584054 |
Roman_2015 |
More_2019, Sahoo_2016, Roman_2015 |
33 |
Šála_2016 |
Purine analogs as phosphatidylinositol 4-kinase IIIβ inhibitors |
Šála, Michal; Kögler, Martin; Plačková, Pavla; Mejdrová, Ivana; Hřebabecký, Hubert; Procházková, Eliška; Strunin, Dmytro; Lee, Gary; Birkus, Gabriel; Weber, Jan; Mertlíková-Kaiserová, Helena; Nencka, Radim |
2016 |
2016-06-01 |
PMC |
N |
PMC7127540 |
27090557.0 |
10.1016/j.bmcl.2016.04.002 |
kifnohj9 |
0.580322 |
|
Im_I_2009, Pérez-Faginas_2011 |
34 |
Kato_2010 |
Development of tetraphenylethylene-based fluorescent oligosaccharide probes for detection of influenza virus |
Kato, Tomohisa; Kawaguchi, Atsushi; Nagata, Kyosuke; Hatanaka, Kenichi |
2010 |
2010-03-26 |
PMC |
N |
PMC7117542 |
20188703.0 |
10.1016/j.bbrc.2010.02.155 |
y9l336oi |
0.579099 |
|
Attioui_1994, Pérez-Faginas_2011, Sahoo_2016 |
35 |
Gürsoy_2020 |
Design and synthesis of novel Imidazo[2,1-b]thiazole derivatives as potent antiviral and antimycobacterial agents |
Gürsoy, Elif; Dincel, Efe Doğukan; Naesens, Lieve; Ulusoy Güzeldemirci, Nuray |
2020 |
2020-01-31 |
PMC |
N |
PMC7112121 |
31862455.0 |
10.1016/j.bioorg.2019.103496 |
c4wnr5xe |
0.577631 |
|
Hamada_2013, Cihan-Üstündağ_2019, Zhao_2016 |
36 |
Singh_2013 |
Regioselective synthesis of 6-substituted-2-amino-5-bromo-4(3H)-pyrimidinones and evaluation of their antiviral activity |
Singh, Kamaljit; Singh, Kawaljit; Balzarini, Jan |
2013 |
2013-09-30 |
PMC |
N |
PMC7127258 |
23911856.0 |
10.1016/j.ejmech.2013.06.036 |
7dxtqde5 |
0.572102 |
|
Paramonova_2017, Pomeisl_2019, Tayade_2015, Głowacka_2015 |
37 |
Mou_J_2009 |
Design, synthesis and primary activity evaluation of l-arginine derivatives as amino-peptidase N/CD13 inhibitors |
Mou, Jiajia; Fang, Hao; Jing, Fanbo; Wang, Qiang; Liu, Yingzi; Zhu, Huawei; Shang, Luqing; Wang, Xuejian; Xu, Wenfang |
2009 |
2009-07-01 |
PMC |
N |
|
19454370.0 |
10.1016/j.bmc.2009.04.056 |
s49954br |
0.563379 |
Ramajayam_2010, Huixiong_Chen_1999, Torres_2012 |
Dude_2008, Konno_2016, Ramajayam_2010 |
38 |
Pahonțu_2015 |
Synthesis, Characterization, Crystal Structure and Antimicrobial Activity of Copper(II) Complexes with the Schiff Base Derived from 2-Hydroxy-4-Methoxybenzaldehyde |
Pahonțu, Elena; Ilieș, Diana-Carolina; Shova, Sergiu; Paraschivescu, Codruța; Badea, Mihaela; Gulea, Aurelian; Roșu, Tudor |
2015 |
2015-04-02 |
COMM-USE |
N |
PMC6272500 |
25849802.0 |
10.3390/molecules20045771 |
0wcvoygd |
0.543965 |
David_2013 |
Sahoo_2016, Zhang_2017, Tabuchi_2009 |
39 |
Pérez-Faginas_2011 |
Synthesis and SAR studies on azetidine-containing dipeptides as HCMV inhibitors |
Pérez-Faginas, Paula; Aranda, M. Teresa; García-López, M. Teresa; Snoeck, Robert; Andrei, Graciela; Balzarini, Jan; González-Muñiz, Rosario |
2011 |
2011-02-01 |
PMC |
N |
PMC7127091 |
21256035.0 |
10.1016/j.bmc.2010.12.052 |
z6ijfhjp |
0.540223 |
|
Cho_A_2012, Im_I_2009, Novikov_2013 |
40 |
Wang_2012 |
First Discovery and Stucture-Activity Relationship Study of Phenanthroquinolizidines as Novel Antiviral Agents against Tobacco Mosaic Virus (TMV) |
Wang, Ziwen; Feng, Anzheng; Cui, Mingbo; Liu, Yuxiu; Wang, Lizhong; Wang, Qingmin |
2012 |
2012-12-28 |
COMM-USE |
N |
PMC3532156 |
23285230.0 |
10.1371/journal.pone.0052933 |
5is9kc52 |
0.533754 |
|
Zhao_2016 |
41 |
Ighilahriz-Boubchir_2017 |
Recyclable Keggin Heteropolyacids as an Environmentally Benign Catalyst for the Synthesis of New 2-Benzoylamino-N-phenyl-benzamide Derivatives under Microwave Irradiations at Solvent-Free Conditions and the Evaluation of Biological Activity |
Ighilahriz-Boubchir, Karima; Boutemeur-Kheddis, Baya; Rabia, Cherifa; Makhloufi-Chebli, Malika; Hamdi, Maamar; Silva, Artur M. S. |
2017 |
2017-12-21 |
COMM-USE |
N |
PMC5943967 |
29267237.0 |
10.3390/molecules23010008 |
h8l7zp2b |
0.531570 |
Mohammat_2009, MacDonald_2012 |
Pahonțu_2015, Pomeisl_2019, Thomson_2010 |
42 |
Zhao_2008 |
Synthesis, cytotoxic activity, and SAR analysis of the derivatives of taxchinin A and brevifoliol |
Zhao, Yu; Guo, Na; Lou, Li-Guang; Cong, Yu-Wen; Peng, Li-Yan; Zhao, Qin-Shi |
2008 |
2008-05-01 |
PMC |
N |
PMC7126827 |
18381240.0 |
10.1016/j.bmc.2008.03.041 |
ur868lpg |
0.531449 |
David_2013 |
Zhang_2018, Carbone_2013, Sahoo_2016 |
43 |
Kuo_R_2009 |
Plant-derived triterpenoids and analogues as antitumor and anti-HIV agents |
Kuo, Reen-Yen; Qian, Keduo; Morris-Natschke, Susan L.; Lee, Kuo-Hsiung |
2009 |
2009-01-01 |
PMC |
N |
PMC3773821 |
19779642.0 |
10.1039/b810774m |
035o1pen |
0.524965 |
|
Ramajayam_2010, Dude_2008, Yadav_2005 |
44 |
Bari_2020 |
Design and syntheses of 7-nitro-2-aryl-4H-benzo[d][1,3]oxazin-4-ones as potent anticancer and antioxidant agents |
Bari, Ayesha; Khan, Zulfiqar Ali; Shahzad, Sohail Anjum; Raza Naqvi, Syed Ali; Khan, Shakeel Ahmad; Amjad, Hira; Iqbal, Ahsan; Yar, Muhammad |
2020 |
2020-08-15 |
PMC |
N |
|
|
10.1016/j.molstruc.2020.128252 |
bow6mfsd |
0.520417 |
Desai_2013 |
Tsoukala_2010, Sahoo_2016, Kumar_2014 |
45 |
Torres_2012 |
Synthesis of benzopolycyclic cage amines: NMDA receptor antagonist, trypanocidal and antiviral activities |
Torres, Eva; Duque, María D.; López-Querol, Marta; Taylor, Martin C.; Naesens, Lieve; Ma, Chunlong; Pinto, Lawrence H.; Sureda, Francesc X.; Kelly, John M.; Vázquez, Santiago |
2012 |
2012-01-15 |
None |
N |
PMC3353318 |
22178660.0 |
10.1016/j.bmc.2011.11.050 |
088gqxyz |
0.504909 |
|
Pérez-Faginas_2011, Cho_A_2012, Głowacka_2015 |
46 |
Zhang_2008 |
Synthesis and in vitro cytotoxicity evaluation of 4-aminoquinoline derivatives |
Zhang, Haiwen; Solomon, V. Raja; Hu, Changkun; Ulibarri, Gerardo; Lee, Hoyun |
2008 |
2008-02-29 |
PMC |
N |
PMC7125724 |
17555912.0 |
10.1016/j.biopha.2007.04.007 |
s1xrwe4h |
0.502459 |
|
Sahoo_2016, Carbone_2013, Zhang_2018 |
47 |
Balzarini_2009 |
Synthesis and anti-HIV studies of 2- and 3-adamantyl-substituted thiazolidin-4-ones |
Balzarini, Jan; Orzeszko-Krzesińska, Barbara; Maurin, Jan K.; Orzeszko, Andrzej |
2009 |
2009-01-31 |
PMC |
N |
PMC7127420 |
18420310.0 |
10.1016/j.ejmech.2008.02.039 |
sw2ufavv |
0.495818 |
Desai_2013, Singh_2013 |
Głowacka_2015, Pomeisl_2019, Carbone_2013, Tsoukala_2010 |
48 |
Jansa_2012 |
An efficient microwave-assisted synthesis and biological properties of polysubstituted pyrimidinyl- and 1,3,5-triazinylphosphonic acids |
Jansa, Petr; Hradil, Ondřej; Baszczyňski, Ondřej; Dračínský, Martin; Klepetářová, Blanka; Holý, Antonín; Balzarini, Jan; Janeba, Zlatko |
2012 |
2012-01-21 |
PMC |
N |
PMC7125588 |
|
10.1016/j.tet.2011.11.040 |
aqezkcyc |
0.492521 |
MacDonald_2012, Yazarians_2017, Mohammat_2009, Nadaraia_2018, Bouton_2017 |
Chopade_2016, Głowacka_2015, Pomeisl_2019, Paramonova_2017, Tsoukala_2010 |
49 |
Zhong_2017 |
Synthesis and biological activity of myricetin derivatives containing 1,3,4-thiadiazole scaffold |
Zhong, Xinmin; Wang, Xiaobin; Chen, Lijuan; Ruan, Xianghui; Li, Qin; Zhang, Juping; Chen, Zhuo; Xue, Wei |
2017 |
2017-10-17 |
COMM-USE |
N |
PMC5645266 |
29086886.0 |
10.1186/s13065-017-0336-7 |
af55iah5 |
0.487317 |
David_2013, Kuo_R_2009 |
Sahoo_2016, Bozorov_2019, Głowacka_2015, Głowacka_2016 |
50 |
Briguglio_2015 |
Benzotriazole: An overview on its versatile biological behavior |
Briguglio, I.; Piras, S.; Corona, P.; Gavini, E.; Nieddu, M.; Boatto, G.; Carta, A. |
2015 |
2015-06-05 |
PMC |
N |
PMC7115563 |
25293580.0 |
10.1016/j.ejmech.2014.09.089 |
aa2taq7z |
0.481915 |
|
Sahoo_2016 |
51 |
Apaydın_2019 |
Synthesis and anti‐coronavirus activity of a series of 1‐thia‐4‐azaspiro[4.5]decan‐3‐one derivatives |
Apaydın, Çağla Begüm; Cesur, Nesrin; Stevaert, Annelies; Naesens, Lieve; Cesur, Zafer |
2019 |
2019-05-09 |
PMC |
N |
PMC7161747 |
31073993.0 |
10.1002/ardp.201800330 |
verzxars |
0.476673 |
|
|
52 |
Kumarasamy_2017 |
Synthesis and in vitro antiviral evaluation of 4-substituted 3,4-dihydropyrimidinones |
Kumarasamy, Dhanabal; Roy, Biswajit Gopal; Rocha-Pereira, Joana; Neyts, Johan; Nanjappan, Satheeshkumar; Maity, Subhasis; Mookerjee, Musfiqua; Naesens, Lieve |
2017 |
2017-01-15 |
PMC |
N |
PMC7127791 |
27979594.0 |
10.1016/j.bmcl.2016.12.010 |
cxpgwwjd |
0.469888 |
|
Cho_A_2012, Hamada_2013, Głowacka_2015 |
53 |
McGuigan_2013 |
Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides |
McGuigan, Christopher; Bourdin, Claire; Derudas, Marco; Hamon, Nadège; Hinsinger, Karen; Kandil, Sahar; Madela, Karolina; Meneghesso, Silvia; Pertusati, Fabrizio; Serpi, Michaela; Slusarczyk, Magdalena; Chamberlain, Stanley; Kolykhalov, Alexander; Vernachio, John; Vanpouille, Christophe; Introini, Andrea; Margolis, Leonid; Balzarini, Jan |
2013 |
2013-12-31 |
None |
N |
PMC4358806 |
24177359.0 |
10.1016/j.ejmech.2013.09.047 |
ziqqalev |
0.461825 |
|
Mehellou_2010, Piotrowska_2019, Hamada_2013, Szűcs_2018 |
54 |
Kaiser_2012 |
A novel type of acyclic nucleoside phosphonates derived from 2-(phosphonomethoxy)propanoic acid |
Kaiser, Martin Maxmilian; Jansa, Petr; Dračínský, Martin; Janeba, Zlatko |
2012 |
2012-05-27 |
PMC |
N |
PMC7111817 |
|
10.1016/j.tet.2012.03.066 |
jcgbotnq |
0.458702 |
Bouton_2017 |
Hocková_2011, Pomeisl_2019, Głowacka_2015, Kasthuri_2011 |
55 |
Raj_R_2014 |
Synthesis and preliminary in vitro activity of mono- and bis-1H-1,2,3-triazole-tethered β-lactam–isatin conjugates against the human protozoal pathogen Trichomonas vaginalis |
Raj, Raghu; Sharma, Vaishali; Hopper, Melissa J.; Patel, Neal; Hall, Dominique; Wrischnik, Lisa A.; Land, Kirkwood M.; Kumar, Vipan |
2014 |
2014-02-22 |
PMC |
N |
PMC7080013 |
|
10.1007/s00044-014-0956-6 |
05jveocv |
0.448984 |
David_2013 |
Tsoukala_2010, Piotrowska_2012, Pomeisl_2019 |
56 |
Yadav_2005 |
Synthesis of 4-hydroxy-1-methylindole and benzo[b]thiophen-4-ol based unnatural flavonoids as new class of antimicrobial agents |
Yadav, Prem P.; Gupta, Prasoon; Chaturvedi, A.K.; Shukla, P.K.; Maurya, Rakesh |
2005 |
2005-03-01 |
PMC |
N |
PMC7125744 |
15698765.0 |
10.1016/j.bmc.2004.12.032 |
hyxj4vgo |
0.446153 |
Kuo_R_2009, Nadaraia_2018, Desai_2013 |
Paramonova_2017, Tayade_2015 |
57 |
Kaur_2017 |
Recent synthetic and medicinal perspectives of dihydropyrimidinones: A review |
Kaur, Ramandeep; Chaudhary, Sandeep; Kumar, Kapil; Gupta, Manish K.; Rawal, Ravindra K. |
2017 |
2017-05-26 |
PMC |
N |
PMC7115489 |
28342939.0 |
10.1016/j.ejmech.2017.03.025 |
bfd5ts44 |
0.440396 |
|
|
58 |
Novikov_2011 |
1-[2-(2-Benzoyl- and 2-benzylphenoxy)ethyl]uracils as potent anti-HIV-1 agents |
Novikov, Mikhail S.; Ivanova, Olga N.; Ivanov, Alexander V.; Ozerov, Alexander A.; Valuev-Elliston, Vladimir T.; Temburnikar, Kartik; Gurskaya, Galina V.; Kochetkov, Sergey N.; Pannecouque, Christophe; Balzarini, Jan; Seley-Radtke, Katherine L. |
2011 |
2011-10-01 |
PMC |
N |
PMC7127633 |
21903401.0 |
10.1016/j.bmc.2011.08.025 |
1nk1trsa |
0.438477 |
|
Głowacka_2015, Paramonova_2017, Tsoukala_2010 |
59 |
Liang_2019 |
Synthesis and structure-activity relationship studies of water-soluble β-cyclodextrin-glycyrrhetinic acid conjugates as potential anti-influenza virus agents |
Liang, Shuobin; Li, Man; Yu, Xiaojuan; Jin, Hongwei; Zhang, Yongmin; Zhang, Lihe; Zhou, Demin; Xiao, Sulong |
2019 |
2019-03-15 |
None |
N |
PMC7115653 |
30731401.0 |
10.1016/j.ejmech.2019.01.074 |
edinv5ou |
0.430476 |
|
Szűcs_2018, Mehellou_2010 |
60 |
Bozorov_2019 |
1,2,3-Triazole-containing hybrids as leads in medicinal chemistry: A recent overview |
Bozorov, Khurshed; Zhao, Jiangyu; Aisa, Haji A. |
2019 |
2019-08-15 |
PMC |
N |
|
31300317.0 |
10.1016/j.bmc.2019.07.005 |
nb73qdix |
0.429108 |
Kuo_R_2009, MacDonald_2012, Mlostoń_2010, Ghosh_2015 |
Kryshchyshyn_2018, Głowacka_2015, Carbone_2013, Sahoo_2016 |
61 |
Pavić_2016 |
Design, Synthesis and Biological Evaluation of Novel Primaquine-Cinnamic Acid Conjugates of the Amide and Acylsemicarbazide Type |
Pavić, Kristina; Perković, Ivana; Gilja, Petra; Kozlina, Filip; Ester, Katja; Kralj, Marijeta; Schols, Dominique; Hadjipavlou-Litina, Dimitra; Pontiki, Eleni; Zorc, Branka |
2016 |
2016-11-28 |
None |
N |
PMC6273687 |
27916811.0 |
10.3390/molecules21121629 |
jmj7se6c |
0.426669 |
David_2013, Rajić_2010 |
Sahoo_2016, Parmenopoulou_2016, Tsoukala_2010 |
62 |
Ghosh_2015 |
Organic Carbamates in Drug Design and Medicinal Chemistry |
Ghosh, Arun K.; Brindisi, Margherita |
2015 |
2015-01-07 |
PMC |
N |
PMC4393377 |
25565044.0 |
10.1021/jm501371s |
o8rlqsq5 |
0.426382 |
Mlostoń_2010, Bozorov_2019 |
Bozorov_2019, Ramajayam_2010, Kryshchyshyn_2018 |
63 |
Jansa_2014 |
5-Substituted 2-amino-4,6-dihydroxypyrimidines and 2-amino-4,6-dichloropyrimidines: synthesis and inhibitory effects on immune-activated nitric oxide production |
Jansa, Petr; Holý, Antonín; Dračínský, Martin; Kolman, Viktor; Janeba, Zlatko; Kostecká, Petra; Kmoníčková, Eva; Zídek, Zdeněk |
2014 |
2014-05-09 |
PMC |
N |
PMC7080047 |
|
10.1007/s00044-014-1018-9 |
kwehwh61 |
0.424305 |
Singh_2013, Mohammat_2009 |
Tsoukala_2010, Manta_2009, Pomeisl_2019 |
64 |
Flütsch_2011 |
HIV-1 protease inhibition potential of functionalized polyoxometalates |
Flütsch, Andreas; Schroeder, Thilo; Grütter, Markus G.; Patzke, Greta R. |
2011 |
2011-02-15 |
None |
N |
PMC7126215 |
21256010.0 |
10.1016/j.bmcl.2010.12.103 |
ieicuxe4 |
0.422071 |
|
|
65 |
Preobrazhenskaya_2006 |
Polycyclic peptide and glycopeptide antibiotics and their derivatives as inhibitors of HIV entry |
Preobrazhenskaya, Maria N.; Olsufyeva, Eugenia N. |
2006 |
2006-09-30 |
PMC |
N |
PMC7114112 |
16720053.0 |
10.1016/j.antiviral.2006.04.008 |
jvqvcz5j |
0.420790 |
|
Lin_J_2008, Szűcs_2018 |
66 |
Bouton_2017 |
Efficient diastereoselective synthesis of a new class of azanucleosides: 2′-homoazanucleosides |
Bouton, Jakob; Van Hecke, Kristof; Van Calenbergh, Serge |
2017 |
2017-07-27 |
PMC |
N |
PMC7111761 |
|
10.1016/j.tet.2017.05.083 |
2a5q6d45 |
0.420716 |
MacDonald_2012, Yang_2008, Yazarians_2017, Yoshizawa_2020 |
Pomeisl_2019, Cho_A_2012, Kaiser_2012 |
67 |
Yang_2009 |
Design and synthesis of novel chloramphenicol amine derivatives as potent aminopeptidase N (APN/CD13) inhibitors |
Yang, Kanghui; Wang, Qiang; Su, Li; Fang, Hao; Wang, Xuejian; Gong, Jianzhi; Wang, Binghe; Xu, Wenfang |
2009 |
2009-06-01 |
PMC |
N |
|
19423354.0 |
10.1016/j.bmc.2009.04.038 |
010lano6 |
0.419223 |
Huixiong_Chen_1999, Ramajayam_2010, Torres_2012, Desai_2013 |
|
68 |
Li_J_2013 |
Epimeric methylsulfinyladenosine derivatives from the marine ascidian Herdmania momus |
Li, Jian Lin; Kim, Eun La; Wang, Haibo; Hong, Jongki; Shin, Sook; Lee, Chong-Kyo; Jung, Jee H. |
2013 |
2013-08-15 |
PMC |
N |
PMC7127152 |
23810281.0 |
10.1016/j.bmcl.2013.05.097 |
o23wv5jw |
0.409273 |
Kuo_R_2009 |
Dude_2008, Almeida_2011 |
69 |
Kumar_2014 |
1H-1,2,3-triazole tethered isatin-ferrocene conjugates: Synthesis and in vitro antimalarial evaluation |
Kumar, Kewal; Pradines, Bruno; Madamet, Marilyn; Amalvict, Rémy; Benoit, Nicolas; Kumar, Vipan |
2014 |
2014-11-24 |
PMC |
N |
PMC7126053 |
25440881.0 |
10.1016/j.ejmech.2014.10.024 |
wc4xirpp |
0.404226 |
Nisha_2014, Singh_2012, Dude_2008, Desai_2013 |
Głowacka_2015, Chopade_2016, Cho_A_2012 |
70 |
Quadrelli_2019 |
Chapter 1 Cycloaddition reactions for antiviral compounds |
Quadrelli, Paolo; Moiola, Mattia |
2019 |
2019-12-31 |
PMC |
N |
PMC7149647 |
|
10.1016/b978-0-12-815273-7.00001-0 |
j7v8g5la |
0.402719 |
MacDonald_2012, Mlostoń_2010, Roman_2015 |
Sahoo_2016, Bozorov_2019, Hamada_2013 |
71 |
Li_W_2008 |
5′-Fluoro-5′-deoxyaristeromycin |
Li, Weikuan; Yin, Xueqiang; Schneller, Stewart W. |
2008 |
2008-01-01 |
None |
N |
PMC2692407 |
18023578.0 |
10.1016/j.bmcl.2007.10.095 |
1g7anngu |
0.393278 |
|
Quintiliani_2011, Pomeisl_2019, Chen_2018, Głowacka_2015 |
72 |
Yates_2019 |
The evolution of antiviral nucleoside analogues: A review for chemists and non-chemists. Part II: Complex modifications to the nucleoside scaffold |
Yates, Mary K.; Seley-Radtke, Katherine L. |
2019 |
2019-02-28 |
PMC |
N |
PMC6349489 |
30529089.0 |
10.1016/j.antiviral.2018.11.016 |
lyq6mec1 |
0.391553 |
|
McGuigan_2013, Hamada_2013 |
73 |
Torres_2014 |
Azapropellanes with Anti-Influenza A Virus Activity |
Torres, Eva; Leiva, Rosana; Gazzarrini, Sabrina; Rey-Carrizo, Matías; Frigolé-Vivas, Marta; Moroni, Anna; Naesens, Lieve; Vázquez, Santiago |
2014 |
2014-05-05 |
PMC |
N |
PMC4094260 |
25050174.0 |
10.1021/ml500108s |
bu9e0twb |
0.388009 |
David_2013 |
Cho_A_2012, Im_I_2009, Pérez-Faginas_2011 |
74 |
Sokolova_2014 |
Camphor-based symmetric diimines as inhibitors of influenza virus reproduction |
Sokolova, Anastasiya S.; Yarovaya, Оlga I.; Korchagina, Dina V.; Zarubaev, Vladimir V.; Tretiak, Tatiana S.; Anfimov, Pavel M.; Kiselev, Oleg I.; Salakhutdinov, Nariman F. |
2014 |
2014-04-01 |
PMC |
N |
PMC7126937 |
24631360.0 |
10.1016/j.bmc.2014.02.038 |
kd6bfps9 |
0.384979 |
|
Tonelli_2017 |
75 |
Pérard-Viret_2017 |
Chapter Four Cephalotaxus Alkaloids |
Pérard-Viret, Joëlle; Quteishat, Laith; Alsalim, Rana; Royer, Jacques; Dumas, Françoise |
2017 |
2017-12-31 |
PMC |
N |
PMC7110560 |
28838429.0 |
10.1016/bs.alkal.2017.07.001 |
m3mhj6op |
0.383107 |
|
Gondim_2019 |
76 |
Duque_2009 |
Synthesis and pharmacological evaluation of (2-oxaadamant-1-yl)amines |
Duque, María D.; Camps, Pelayo; Profire, Lenuta; Montaner, Silvia; Vázquez, Santiago; Sureda, Francesc X.; Mallol, Jordi; López-Querol, Marta; Naesens, Lieve; Clercq, Erik De; Radhika Prathalingam, S.; Kelly, John M. |
2009 |
2009-04-15 |
None |
N |
PMC3217223 |
19251424.0 |
10.1016/j.bmc.2009.02.007 |
x7s1f9gd |
0.383041 |
Torres_2012 |
Paramonova_2017, Ramajayam_2010, Cho_A_2012 |
77 |
Konno_2016 |
Design and synthesis of a series of serine derivatives as small molecule inhibitors of the SARS coronavirus 3CL protease |
Konno, Hiroyuki; Wakabayashi, Masaki; Takanuma, Daiki; Saito, Yota; Akaji, Kenichi |
2016 |
2016-03-15 |
PMC |
N |
PMC7111485 |
26879854.0 |
10.1016/j.bmc.2016.01.052 |
9bw1z5ps |
0.376168 |
Ramajayam_2010, Regnier_2009, Ramajayam_2010 |
Dude_2008, Im_I_2009, Ramajayam_2010, Chen_2005 |
78 |
Thanigaimalai_2013 |
Development of potent dipeptide-type SARS-CoV 3CL protease inhibitors with novel P3 scaffolds: Design, synthesis, biological evaluation, and docking studies |
Thanigaimalai, Pillaiyar; Konno, Sho; Yamamoto, Takehito; Koiwai, Yuji; Taguchi, Akihiro; Takayama, Kentaro; Yakushiji, Fumika; Akaji, Kenichi; Chen, Shen-En; Naser-Tavakolian, Aurash; Schön, Arne; Freire, Ernesto; Hayashi, Yoshio |
2013 |
2013-10-31 |
None |
N |
PMC7115411 |
23994330.0 |
10.1016/j.ejmech.2013.07.037 |
olfpcndb |
0.374492 |
|
Konno_2013, Thanigaimalai_2013 |
79 |
Egan_2004 |
Potent antiviral agent WIN 54954: high specific activity labelling with tritium |
Egan, Judith A.; Nugent, Richard P.; Filer, Crist N. |
2004 |
2004-06-30 |
PMC |
N |
PMC7127203 |
15110350.0 |
10.1016/j.apradiso.2004.03.002 |
8dqniuzd |
0.371042 |
David_2013 |
Dude_2008 |
80 |
Nisha_2014 |
N-Propargylated isatin-Mannich mono- and bis-adducts: Synthesis and preliminary analysis of in vitro activity against Tritrichomonas foetus |
Nisha, ; Kumar, Kewal; Bhargava, Gaurav; Land, Kirkwood M.; Chang, Kai-Hsiang; Arora, Reena; Sen, Somdutta; Kumar, Vipan |
2014 |
2014-03-03 |
PMC |
N |
PMC7115568 |
24561663.0 |
10.1016/j.ejmech.2014.01.015 |
hzfawetp |
0.368174 |
|
Kumar_2014, Raj_R_2014, Chopade_2016 |
81 |
Karaküçük-İyidoğan_2019 |
Synthesis, Biological Evaluation and Ligand Based Pharmacophore Modeling of New Aromatic Thiosemicarbazones as Potential Anticancer Agents |
Karaküçük-İyidoğan, A.; Aydınöz, B.; Taşkın-Tok, T.; Oruç-Emre, E. E.; Balzarini, J. |
2019 |
2019-05-15 |
PMC |
N |
PMC7089137 |
|
10.1007/s11094-019-01968-3 |
jyti99xq |
0.365412 |
|
Piotrowska_2019, Sahoo_2016, Hamada_2013, McGuigan_2013 |
82 |
Zhao_2020 |
Pyrazolone structural motif in medicinal chemistry: Retrospect and prospect |
Zhao, Zefeng; Dai, Xufen; Li, Chenyang; Wang, Xiao; Tian, Jiale; Feng, Ying; Xie, Jing; Ma, Cong; Nie, Zhuang; Fan, Peinan; Qian, Mingcheng; He, Xirui; Wu, Shaoping; Zhang, Yongmin; Zheng, Xiaohui |
2020 |
2020-01-15 |
PMC |
N |
PMC7115706 |
31761383.0 |
10.1016/j.ejmech.2019.111893 |
qxbdr377 |
0.363861 |
|
|
83 |
Olsufyeva_2020 |
Main trends in the design of semi-synthetic antibiotics of a new generation |
Olsufyeva, Evgenia N.; Yankovskaya, Valentina S. |
2020 |
2020-03-23 |
PMC |
N |
PMC7149660 |
|
10.1070/rcr4892 |
nypnib0h |
0.360275 |
|
Zhao_2016 |
84 |
Baltina_2015 |
Glycyrrhizic acid derivatives as influenza A/H1N1 virus inhibitors |
Baltina, Lidia A.; Zarubaev, Vladimir V.; Baltina, Lia A.; Orshanskaya, Iana A.; Fairushina, Alina I.; Kiselev, Oleg I.; Yunusov, Marat S. |
2015 |
2015-04-15 |
PMC |
N |
PMC7127794 |
25801933.0 |
10.1016/j.bmcl.2015.02.074 |
d6do1xad |
0.359257 |
Lin_D_2012 |
Lin_J_2008, Pérez-Faginas_2011 |
85 |
Siebert_2018 |
Synthesis and antimicrobial activity of amino acid and peptide derivatives of mycophenolic acid |
Siebert, Agnieszka; Wysocka, Magdalena; Krawczyk, Beata; Cholewiński, Grzegorz; Rachoń, Janusz |
2018 |
2018-01-01 |
PMC |
N |
|
29216563.0 |
10.1016/j.ejmech.2017.11.094 |
wydc0wyd |
0.359145 |
|
|
86 |
Kim_M_2011 |
2,6-Bis-arylmethyloxy-5-hydroxychromones with antiviral activity against both hepatitis C virus (HCV) and SARS-associated coronavirus (SCV) |
Kim, Mi Kyoung; Yu, Mi-Sun; Park, Hye Ri; Kim, Kyung Bo; Lee, Chaewoon; Cho, Suh Young; Kang, Jihoon; Yoon, Hyunjun; Kim, Dong-Eun; Choo, Hyunah; Jeong, Yong-Joo; Chong, Youhoon |
2011 |
2011-11-30 |
PMC |
N |
PMC7115508 |
21925774.0 |
10.1016/j.ejmech.2011.09.005 |
garchpin |
0.352463 |
|
Mehellou_2010, Ikejiri_2007, Tsoukala_2010 |
87 |
Kang_2016 |
First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via ‘privileged scaffold’ refining approach |
Kang, Dongwei; Zhang, Heng; Zhou, Zhongxia; Huang, Boshi; Naesens, Lieve; Zhan, Peng; Liu, Xinyong |
2016 |
2016-11-01 |
PMC |
N |
PMC7126219 |
27742238.0 |
10.1016/j.bmcl.2016.09.071 |
8yhsjbmi |
0.347592 |
|
Tsoukala_2010, Piotrowska_2012, Głowacka_2015 |
88 |
Macan_2019 |
Antitumor and antiviral activities of 4-substituted 1,2,3-triazolyl-2,3-dibenzyl-L-ascorbic acid derivatives |
Macan, Andrijana Meščić; Harej, Anja; Cazin, Ines; Klobučar, Marko; Stepanić, Višnja; Pavelić, Krešimir; Pavelić, Sandra Kraljević; Schols, Dominique; Snoeck, Robert; Andrei, Graciela; Raić-Malić, Silvana |
2019 |
2019-12-15 |
PMC |
N |
PMC7115614 |
31586832.0 |
10.1016/j.ejmech.2019.111739 |
4w0zw3br |
0.347252 |
|
Głowacka_2015, Tsoukala_2010, Piotrowska_2012 |
89 |
Song_2012 |
Synthesis and Biochemical Evaluation of Thiochromanone Thiosemicarbazone Analogues as Inhibitors of Cathepsin L |
Song, Jiangli; Jones, Lindsay\nM.; Kumar, G. D. Kishore; Conner, Elizabeth S.; Bayeh, Liela; Chavarria, Gustavo E.; Charlton-Sevcik, Amanda K.; Chen, Shen-En; Chaplin, David J.; Trawick, Mary Lynn; Pinney, Kevin G. |
2012 |
2012-04-30 |
PMC |
N |
PMC4025852 |
24900494.0 |
10.1021/ml200299g |
qqhkc3f1 |
0.343509 |
Ramajayam_2010, Huixiong_Chen_1999, Kishore_Kumar_2010 |
Kishore_Kumar_2010, Sahoo_2016, Piotrowska_2019 |
90 |
Zhong_2015 |
Discovery of Metal Ions Chelator Quercetin Derivatives with Potent Anti-HCV Activities |
Zhong, Dongwei; Liu, Mingming; Cao, Yang; Zhu, Yelin; Bian, Shihui; Zhou, Jiayi; Wu, Fengjie; Ryu, Kum-Chol; Zhou, Lu; Ye, Deyong |
2015 |
2015-04-16 |
COMM-USE |
N |
PMC6272327 |
25913935.0 |
10.3390/molecules20046978 |
rhld75dy |
0.342252 |
|
Sahoo_2016, Lin_J_2008 |
91 |
Khandaker_2019 |
Synthesis and Evaluations of “1,4‐Triazolyl Combretacoumarins” and Desmethoxy Analogs |
Khandaker, Tashrique A.; Hess, Jessica D.; Aguilera, Renato; Andrei, Graciela; Snoeck, Robert; Schols, Dominique; Pradhan, Padmanava; Lakshman, Mahesh K. |
2019 |
2019-08-07 |
PMC |
N |
PMC6774347 |
31579393.0 |
10.1002/ejoc.201900569 |
90pat7ij |
0.338308 |
|
|
92 |
Kaminskyy_2017 |
5-Ene-4-thiazolidinones – An efficient tool in medicinal chemistry |
Kaminskyy, Danylo; Kryshchyshyn, Anna; Lesyk, Roman |
2017 |
2017-11-10 |
PMC |
N |
PMC7111298 |
28987611.0 |
10.1016/j.ejmech.2017.09.031 |
nzykgiyr |
0.334748 |
|
Carbone_2013, Bozorov_2019, Kryshchyshyn_2018, Sahoo_2016 |
93 |
Ben_Salem_2011 |
Molecular drug-organiser: Synthesis, characterization and biological evaluation of penicillin V and/or nalidixic acid calixarene-based podands |
Ben Salem, Adel; Sautrey, Guillaume; Fontanay, Stéphane; Duval, Raphaël E.; Regnouf-de-Vains, Jean-Bernard |
2011 |
2011-12-15 |
PMC |
N |
|
22075235.0 |
10.1016/j.bmc.2011.10.031 |
ws07d3ti |
0.331146 |
Siebert_2018 |
Szűcs_2018, Sahoo_2016 |
94 |
Lyakhova_2009 |
Synthesis and affinity to DNA of phenylbenzoimidazoles and benzoimidazo[1,2-c]quinazolines |
Lyakhova, Elena A.; Gusyeva, Yulia A.; Nekhoroshkova, Julia V.; Shafran, Lev M.; Lyakhov, Sergey A. |
2009 |
2009-08-31 |
PMC |
N |
PMC7115644 |
19349097.0 |
10.1016/j.ejmech.2009.03.004 |
t19szy8k |
0.329038 |
|
Głowacka_2015, Paramonova_2017, Cho_A_2012 |
95 |
Kabir_2008 |
New classes of Gram-positive selective antibacterials: Inhibitors of MRSA and surrogates of the causative agents of anthrax and tuberculosis |
Kabir, M. Shahjahan; Engelbrecht, Kathleen; Polanowski, Rebecca; Krueger, Sarah M.; Ignasiak, Rachel; Rott, Marc; Schwan, William R.; Stemper, Mary E.; Reed, Kurt D.; Sherman, David; Cook, James M.; Monte, Aaron |
2008 |
2008-11-01 |
PMC |
N |
PMC7127099 |
18849164.0 |
10.1016/j.bmcl.2008.09.085 |
8zmlqdc1 |
0.328424 |
Siebert_2018 |
Zhao_2016, Opsenica_2011 |
96 |
Ye_N_2015 |
Structure–Activity Relationship Studies of Substituted 2-(Isoxazol-3-yl)-2-oxo-N′-phenyl-acetohydrazonoyl Cyanide Analogues: Identification of Potent Exchange Proteins Directly Activated by cAMP (EPAC) Antagonists |
Ye, Na; Zhu, Yingmin; Chen, Haijun; Liu, Zhiqing; Mei, Fang C.; Wild, Christopher; Chen, Haiying; Cheng, Xiaodong; Zhou, Jia |
2015 |
2015-07-16 |
PMC |
N |
PMC4769034 |
26151319.0 |
10.1021/acs.jmedchem.5b00635 |
3yk35rr0 |
0.325259 |
|
Deiab_2015 |
97 |
Cihan-Üstündağ_2019 |
Design, synthesis, antitubercular and antiviral properties of new spirocyclic indole derivatives |
Cihan-Üstündağ, Gökçe; Naesens, Lieve; Şatana, Dilek; Erköse-Genç, Gonca; Mataracı-Kara, Emel; Çapan, Gültaze |
2019 |
2019-07-17 |
PMC |
N |
PMC7087588 |
|
10.1007/s00706-019-02457-9 |
cu1uprwm |
0.324818 |
David_2013 |
Zhao_2016, Hamada_2013, Cihan-Üstündağ_2016 |
98 |
Musella_2016 |
Identification of an indol-based derivative as potent and selective varicella zoster virus (VZV) inhibitor |
Musella, Simona; di Sarno, Veronica; Ciaglia, Tania; Sala, Marina; Spensiero, Antonia; Scala, Maria Carmina; Ostacolo, Carmine; Andrei, Graciela; Balzarini, Jan; Snoeck, Robert; Novellino, Ettore; Campiglia, Pietro; Bertamino, Alessia; Gomez-Monterrey, Isabel M. |
2016 |
2016-11-29 |
PMC |
N |
PMC7115581 |
27639368.0 |
10.1016/j.ejmech.2016.09.014 |
gnnis7pl |
0.323820 |
|
Lin_J_2008, Opsenica_2011 |
99 |
El-Faham_2015 |
Synthesis, Characterization, and Anti-Cancer Activity of Some New N′-(2-Oxoindolin-3-ylidene)-2-propylpentane hydrazide-hydrazones Derivatives |
El-Faham, Ayman; Farooq, Muhammad; Khattab, Sherine N.; Abutaha, Nael; Wadaan, Mohammad A.; Ghabbour, Hazem A.; Fun, Hoong-Kun |
2015 |
2015-08-13 |
COMM-USE |
N |
PMC6332339 |
26287132.0 |
10.3390/molecules200814638 |
0dddrh4e |
0.321290 |
David_2013 |
Carbone_2013, Tsoukala_2010, Głowacka_2015 |
100 |
Ikejiri_2007 |
Synthesis and biological evaluation of nucleoside analogues having 6-chloropurine as anti-SARS-CoV agents |
Ikejiri, Masahiro; Saijo, Masayuki; Morikawa, Shigeru; Fukushi, Shuetsu; Mizutani, Tetsuya; Kurane, Ichiro; Maruyama, Tokumi |
2007 |
2007-05-01 |
PMC |
N |
PMC7126875 |
17336519.0 |
10.1016/j.bmcl.2007.02.026 |
nltbvlzq |
0.316705 |
Novikov_2011, Shin_2018 |
Pérez-Faginas_2011, Cho_A_2012, Ramajayam_2010 |
101 |
Yoon_2019 |
Study on the 2‐Phenylchroman‐4‐One Derivatives and their anti‐MERS‐CoV Activities |
Yoon, Ji Hye; Lee, Jihye; Lee, Jun Young; Shin, Young Sup; Kim, Dong Eon; Min, Jung Sun; Park, Chul Min; Song, Jong Hwan; Kim, Seungtaek; Kwon, Sunoh; Jang, Min Seong; Kim, Hyoung Rae |
2019 |
2019-07-28 |
PMC |
N |
PMC7161870 |
|
10.1002/bkcs.11832 |
qg3hl5ft |
0.314587 |
Hjortland_2016 |
|
102 |
Wang_2018 |
Structure-activity relationships of cryptopleurine analogs with E-ring modifications as anti-hepatitis C virus agents |
Wang, Ying; Chen, Shao-Ru; Yang, Xiaoming; Lee, Kuo-Hsiung; Cheng, Yung-Chi |
2018 |
2018-02-01 |
PMC |
N |
|
29317151.0 |
10.1016/j.bmc.2017.12.027 |
9vssue3m |
0.314305 |
|
|
103 |
Rachwal_2008 |
5.01 1,2,3-Triazoles |
Rachwal, S.; Katritzky, A.R. |
2008 |
2008-12-31 |
PMC |
N |
|
|
10.1016/b978-008044992-0.00501-0 |
qobzttqa |
0.313359 |
|
Bozorov_2019, Pomeisl_2019, Głowacka_2015 |
104 |
Roman_2015 |
Mannich bases in medicinal chemistry and drug design |
Roman, Gheorghe |
2015 |
2015-01-07 |
PMC |
N |
PMC7115492 |
25462280.0 |
10.1016/j.ejmech.2014.10.076 |
f8pyn3rx |
0.307436 |
|
|
105 |
Yadav_2019 |
Synthetic, Structural, and Anticancer Activity Evaluation Studies on Novel Pyrazolylnucleosides |
Yadav, Yogesh; Sharma, Deepti; Kaushik, Kumar; Kumar, Vineet; Jha, Amitabh; Prasad, Ashok K.; Len, Christophe; Malhotra, Sanjay V.; Wengel, Jesper; Parmar, Virinder S. |
2019 |
2019-10-30 |
COMM-USE |
N |
PMC6864788 |
31671703.0 |
10.3390/molecules24213922 |
15rg623y |
0.307198 |
David_2013 |
Desai_2013, Li_Y_2016, Kumarasamy_2017, Carbone_2013 |
106 |
Wang_2017 |
Discovery of unsymmetrical aromatic disulfides as novel inhibitors of SARS-CoV main protease: Chemical synthesis, biological evaluation, molecular docking and 3D-QSAR study |
Wang, Li; Bao, Bo-Bo; Song, Guo-Qing; Chen, Cheng; Zhang, Xu-Meng; Lu, Wei; Wang, Zefang; Cai, Yan; Li, Shuang; Fu, Sheng; Song, Fu-Hang; Yang, Haitao; Wang, Jian-Guo |
2017 |
2017-09-08 |
PMC |
N |
PMC7115414 |
28624700.0 |
10.1016/j.ejmech.2017.05.045 |
mxnx4mmu |
0.306697 |
|
Liu_W_2014, Thanigaimalai_2013 |
107 |
Khanna_2020 |
Spiro‐Indole‐Coumarin Hybrids: Synthesis, ADME, DFT, NBO Studies and In Silico Screening through Molecular Docking on DNA G‐Quadruplex |
Khanna, Leena; Singhal, Sugandha; Jain, Subhash C.; Khanna, Pankaj |
2020 |
2020-03-19 |
PMC |
N |
PMC7169502 |
|
10.1002/slct.201904783 |
5drr3fyt |
0.306514 |
|
|
108 |
Xu_J_2010 |
QSAR Studies on Andrographolide Derivatives as α-Glucosidase Inhibitors |
Xu, Jun; Huang, Sichao; Luo, Haibin; Li, Guoji; Bao, Jiaolin; Cai, Shaohui; Wang, Yuqiang |
2010 |
2010-03-02 |
COMM-USE |
N |
PMC2869241 |
20479989.0 |
10.3390/ijms11030880 |
s0ps9rd0 |
0.306370 |
|
Zhong_2015, Li_X_2019 |
109 |
Konno_2017 |
Synthesis and evaluation of phenylisoserine derivatives for the SARS-CoV 3CL protease inhibitor |
Konno, Hiroyuki; Onuma, Takumi; Nitanai, Ikumi; Wakabayashi, Masaki; Yano, Shigekazu; Teruya, Kenta; Akaji, Kenichi |
2017 |
2017-06-15 |
PMC |
N |
PMC7127027 |
28454669.0 |
10.1016/j.bmcl.2017.04.056 |
qym6jch0 |
0.302802 |
Ramajayam_2010 |
Ramajayam_2010, Konno_2016, Dude_2008, Konno_2013 |
110 |
Ouahrouch_2015 |
Design, Synthesis, and Antiviral Activity of Novel Ribonucleosides of 1,2,3‐Triazolylbenzyl‐aminophosphonates |
Ouahrouch, Abdelaaziz; Taourirte, Moha; Schols, Dominique; Snoeck, Robert; Andrei, Graciela; Engels, Joachim W.; Lazrek, Hassan B. |
2015 |
2015-11-17 |
NONCOMM |
N |
PMC4832832 |
26575425.0 |
10.1002/ardp.201500292 |
25dwlzpy |
0.301550 |
David_2013 |
Głowacka_2015, Cho_A_2012, Kumarasamy_2017 |
111 |
Shimano_1996 |
Synthesis of both enantiomers of halitunal |
Shimano, Kazunori; Ge, Yuting; Sakaguchi, Kazuhiko; Isoe, Sachihiko |
1996 |
1996-03-25 |
PMC |
N |
|
|
10.1016/0040-4039(96)00268-7 |
uhi4vd3a |
0.300287 |
MacDonald_2012, Kuo_R_2009, Mohammat_2009, Nadaraia_2018 |
Lin_Z_2012, Duque_2009, Paramonova_2017, Kasthuri_2011 |
112 |
Attioui_1994 |
Recognition ability and cytotoxicity of some oligosaccharidylsubstituted β-cyclodextrins |
Attioui, Fatima; Al-Omar, Anouar; Leray, Eric; Parrot-Lopez, Hélène; Finance, Chantal; Bonaly, Roger |
1994 |
1994-12-31 |
PMC |
N |
PMC7131397 |
7606211.0 |
10.1016/s0248-4900(94)80018-9 |
vtctnqki |
0.300055 |
|
|